Explore advanced quantitative methodologies shaping modern drug discovery in “Drug Design Strategies: Quantitative Approaches.” This essential guide, curated by leading experts, details how numerical analysis and computational tools, from structure-based design to bioinformatics, enable robust predictions. Discover historical development, current state-of-the-art techniques, and practical examples covering quantitative structure-activity relationships (QSAR), molecular modeling, cheminformatics, and predictive toxicology. Learn to manage chemical structures, assess predictive model quality, and optimize potency, selectivity, ADMET properties, and chemical library design. Ideal for drug design practitioners seeking to enhance efficiency, reduce costs, and shift the balance towards successful drug discovery through rigorous quantitative methods. A must-have resource for improving lead generation and optimization.